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TargetCarbonic anhydrase 2
LigandBDBM50428474
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1554922
Ki 3100000±n/a nM
Citation Vullo, DDel Prete, SDe Luca, VCarginale, VFerraroni, MDedeoglu, NOsman, SMAlOthman, ZCapasso, CSupuran, CT Anion inhibition studies of the฿-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. Bioorg Med Chem Lett26:1406-10 (2016) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Carbonic anhydrase 2
Name:Carbonic anhydrases; II & IX
Synonyms:CA-II | CA2 | CAC | Carbonate dehydratase II | Carbonic anhydrase 2 (CA II) | Carbonic anhydrase 2 (CA-II) | Carbonic anhydrase 2 (Recombinant CA II) | Carbonic anhydrase C | Carbonic anhydrase II (CA II) | Carbonic anhydrase II (CA-II) | Carbonic anhydrase II (CAII) | Carbonic anhydrase II (hCA II) | Carbonic anhydrase isoenzyme II (hCA II)
Type:Enzyme
Mol. Mass.:29250.71
Organism:Homo sapiens (Human)
Description:P00918
Residue:260
Sequence:
MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRIL
NNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHL
VHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDP
RGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELM
VDNWRPAQPLKNRQIKASFK
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BDBM50428474
NameBDBM50428474
Synonyms:DITIOCARB | Diethyldithiocarbamate
TypeSmall organic molecule
Emp. Form.C5H11NS2
Mol. Mass.149.278
SMILESCCN(CC)C(S)=S
Structure
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