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Target
Putative P2Y purinoceptor 10
Ligand
BDBM50177150
Substrate
n/a
Meas. Tech.
ChEMBL_1581711 (CHEMBL3816044)
EC50
17±n/a nM
Citation
 Jung, S; Inoue, A; Nakamura, S; Kishi, T; Uwamizu, A; Sayama, M; Ikubo, M; Otani, Y; Kano, K; Makide, K; Aoki, J; Ohwada, T Conformational Constraint of the Glycerol Moiety of Lysophosphatidylserine Affords Compounds with Receptor Subtype Selectivity. J Med Chem 59:3750-76 (2016) [PubMed]  Article 
Target
Name:
Putative P2Y purinoceptor 10
Synonyms:
P2Y10 | P2Y10_MOUSE | P2ry10 | Putative P2Y purinoceptor 10
Type:
PROTEIN
Mol. Mass.:
37264.07
Organism:
Mus musculus
Description:
ChEMBL_109764
Residue:
328
Sequence:
MGSNSTSSAESNCNATYLPFQYSLYATTYIFIFIPGLLANSAALWVLCRFISKKNKAIIFMINLSVADLAHILSLPLRIYYYINRHWPFQRALCLLCFYLKYLNMYASIFFLTCISLQRCLFLLKPFRARNWKRRYDVGISAVIWIVVGTACLPFPILRNAGLANSTDSCFADLGYKQMDAVVLVTMVVIAELAGFVIPVITIACCTWKTTVSLKHPPIAFQGISERKKALRMVFMCAAVFVICFTPYHINFIFYTMVKESIITSCPTVKSTLYFHPFSLCLASLCCLLDPILYYFMASEFRDQLSRHGSSVTRSRLMSRESGSSMVN
  
Inhibitor
Name:
BDBM50177150
Synonyms:
CHEMBL3813843
Type:
Small organic molecule
Emp. Form.:
C29H46NO10P
Mol. Mass.:
599.65
SMILES:
CCCCCCCCCCCOc1ccccc1CCC(=O)OC[C@H]1OCC=C[C@@H]1OP(O)(=O)OC[C@H](N)C(O)=O |r,c:28|
Structure:
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