Reaction Details Report a problem with these data
Target
Melatonin receptor type 1C
Ligand
BDBM50212914
Substrate
n/a
Meas. Tech.
ChEMBL_104753 (CHEMBL712436)
Ki
27±n/a nM
Citation
  TBA Bioorg Med Chem Lett 4:1555-1558 (1994)   
Target
Name:
Melatonin receptor type 1C
Synonyms:
CKB | MTR1C_CHICK | Mel-1C-R | Mel1c receptor | Melatonin receptor type 1C
Type:
PROTEIN
Mol. Mass.:
38595.98
Organism:
Gallus gallus
Description:
ChEMBL_104739
Residue:
346
Sequence:
MERPGSNGSCSGCRLEGGPAARAASGLAAVLIVTIVVDVLGNALVILSVLRNKKLRNAGNIFVVSLSVADLVVAVYPYPLILSAIFHNGWTMGNIHCQISGFLMGLSVIGSIFNITAIAINRYCYICHSLRYDKLFNLKNTCCYICLTWTLTVVAIVPNFFVGSLQYDPRIYSCTFAQTVSTSYTITVVVVHFIVPLSIVTFCYLRIWILVIQVKHRVRQDCKQKIRAADIRNFLTMFVVFVLFAVCWGPLNFIGLAVSINPSKVQPHIPEWLFVLSYFMAYFNSCLNAVIYGLLNQNFRKEYKRILLMLRTPRLLFIDVSKGGTEGLKSKPSPAVTNNNQAEIHL
  
Inhibitor
Name:
BDBM50212914
Synonyms:
CHEMBL39667
Type:
Small organic molecule
Emp. Form.:
C13H14Br2N2O
Mol. Mass.:
374.071
SMILES:
CCC(=O)NCCc1c(Br)[nH]c2cc(Br)ccc12
Structure:
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