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Target
Substance-K receptor
Ligand
BDBM84953
Substrate
n/a
Ki
8.4±n/a nM
Comments
PDSP_1176
Citation
Kudlacz, EM; Shatzer, SA; Knippenberg, RW; Logan, DE; Poirot, M; van Giersbergen, PL; Burkholder, TP In vitro and in vivo characterization of MDL 105,212A, a nonpeptide NK-1/NK-2 tachykinin receptor antagonist. J Pharmacol Exp Ther 277:840-51 (1996) [PubMed]
More Info.:
Target
Name:
Substance-K receptor
Synonyms:
NK-2 receptor | NK-2R | NK2R_BOVIN | Neurokinin 2 receptor | Neurokinin A receptor | SKR | Substance-K receptor | TAC2R | TACR2 | Tachykinin receptor 2
Type:
PROTEIN
Mol. Mass.:
43078.78
Organism:
Bos taurus
Description:
ChEMBL_143050
Residue:
384
Sequence:
MGACVVMTDINISSGLDSNATGITAFSMPGWQLALWTAAYLALVLVAVMGNATVIWIILAHQRMRTVTNYFIVNLALADLCMAAFNAAFNFVYASHNIWYFGRAFCYFQNLFPITAMFVSIYSMTAIAADRYMAIVHPFQPRLSAPGTRAVIAGIWLVALALAFPQCFYSTITTDEGATKCVVAWPEDSGGKMLLLYHLIVIALIYFLPLVVMFVAYSVIGLTLWRRSVPGHQAHGANLRHLQAKKKFVKTMVLVVVTFAICWLPYHLYFILGTFQEDIYCHKFIQQVYLALFWLAMSSTMYNPIIYCCLNHRFRSGFRLAFRCCPWVTPTEEDKMELTYTPSLSTRVNRCHTKEIFFMSGDVAPSEAVNGQAESPQAGVSTEP