Reaction Details Report a problem with these data
Target
Cholecystokinin
Ligand
BDBM84994
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_1422
Citation
 Schotte, A; Janssen, PF; Gommeren, W; Luyten, WH; Van Gompel, P; Lesage, AS; De Loore, K; Leysen, JE Risperidone compared with new and reference antipsychotic drugs: in vitro and in vivo receptor binding. Psychopharmacology (Berl) 124:57-73 (1996) [PubMed]  Article 
Target
Name:
Cholecystokinin
Synonyms:
CCK | CCKN_PIG | Cholecystokinin B
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12528.64
Organism:
GUINEA PIG
Description:
Cholecystokinin B 0 GUINEA PIG::P01356
Residue:
114
Sequence:
MNGGLCLCVLMAVLAAGTLAQPVPPADSAVPGAQEEEAHRRQLRAVQKVDGESRAHLGALLARYIQQARKAPSGRVSMIKNLQSLDPSHRISDRDYMGWMDFGRRSAEEYEYTS
  
Inhibitor
Name:
BDBM84994
Synonyms:
CAS_163091 | NSC_163091 | ORG-5222
Type:
Small organic molecule
Emp. Form.:
C17H16ClNO
Mol. Mass.:
285.768
SMILES:
CN1CC2C(C1)c1cc(Cl)ccc1Oc1ccccc21
Structure:
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