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Target
CB1 cannabinoid receptor-interacting protein 1
Ligand
BDBM21281
Substrate
n/a
Ki
58.6±n/a nM
Comments
PDSP_1966
Citation
 Stefano, GB; Salzet, B; Salzet, M Identification and characterization of the leech CNS cannabinoid receptor: coupling to nitric oxide release. Brain Res 753:219-24 (1997) [PubMed]  Article 
Target
Name:
CB1 cannabinoid receptor-interacting protein 1
Synonyms:
CANNABINOID CB1 | CNR1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
22425.67
Organism:
theromyzon Tessulatum
Description:
CANNABINOID CB1 CNR1 theromyzon Tessulatum::A0A0V1DID4
Residue:
196
Sequence:
MDTMTMETLLLSSTLLLLPFNKHGGAKLAGWLVNDLPRRRIMKPPSRFEVHIRFCCLKPENAETTFKVDGRRFNMSTKTLKLYRDTTYRIGVTSSPPMEFEEAEINGENLISHLEPDGGIEADWSTAGFSKTKSRSRCNIRLMLRGVFGSVTQDLQCKFYDISDPHAQWGDKFRQMVLVCSTYDDCMINVVEVELK
  
Inhibitor
Name:
BDBM21281
Synonyms:
(11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphthalen-1-ylcarbonyl)-9-oxa-1-azatricyclo[6.3.1.0^{4,12}]dodeca-2,4(12),5,7-tetraene | (2,3-dihydro-5-methyl-3-((4-morpholinyl)methyl)pyrrolo-(1,2,3-de)-1,4-benzoxazin-6-yl)(1-naphthalenyl)methanone monomethanesulfonat | CHEMBL188 | WIN 55,212-2 | WIN 55212-2 | WIN-55212 | WIN55212-2
Type:
Analgesic
Emp. Form.:
C27H26N2O3
Mol. Mass.:
426.5069
SMILES:
Cc1c(C(=O)c2cccc3ccccc23)c2cccc3OC[C@@H](CN4CCOCC4)n1c23 |r|
Structure:
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