Reaction Details Report a problem with these data
Target
Histamine H2 receptor
Ligand
BDBM82472
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_456
Citation
Kennett, GA; Ainsworth, K; Trail, B; Blackburn, TP BW 723C86, a 5-HT2B receptor agonist, causes hyperphagia and reduced grooming in rats. Neuropharmacology 36:233-9 (1997) [PubMed] Article
More Info.:
Target
Name:
Histamine H2 receptor
Synonyms:
HISTAMINE H2 | HRH2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40972.37
Organism:
RABBIT
Description:
HISTAMINE H2 HRH2 RABBIT::G1TWL8
Residue:
367
Sequence:
MEPNDTANDTASSSCLESTAFKVTLSVVLTILILITAAGNVVVCLAVGLNRRLRSLTNCFIVSLAITDLLLGLLVLPFSAIYQLSCRWSFGKVFCNIYISLDVMLCTASILNLFMISIDRYCAVTDPLRYPVLVTPGRVTISLVSIWVISITLSFLSIHLGWNSRNTTSEGHHTSPKCKFQVNEVYGLVDGLVTFYLPLLIMCVTYYRIFKIAREQARRINHISSWQAATIREHKATVTLAAVMGAFIVCWFPYFTTFVYRGLKGDDAINEVVEAVVLWLGYANSALNPILYAALNRDFRNAYQQLFCCRLAGRGSHETCLRFNNALLPKSQSQEPRRQEEKPLKLQVWSGTEATAPQGATDRVFGE