Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 3A
Ligand
BDBM82517
Substrate
n/a
Ki
316±n/a nM
Comments
PDSP_1289
Citation
Mos, J; Van Hest, A; Van Drimmelen, M; Herremans, AH; Olivier, B The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons. Eur J Pharmacol 325:145-53 (1997) [PubMed] Article
More Info.:
Target
Name:
5-hydroxytryptamine receptor 3A
Synonyms:
5-HT3 | HTR3A
Type:
Enzyme Catalytic Domain
Mol. Mass.:
46633.35
Organism:
pigeon
Description:
5-HT3 HTR3A pigeon::A0A218UVI3
Residue:
407
Sequence:
MIGILFPAGAAPKYLCTYYDIVDYLNISSHDKLHTYILPKKDLQEPVEVTMDFFLVAILSVVEKLQTVSFYFVLNLEWQNPFATWNPRDFCNISEIVLPMDTYWSPPIFFLERVNGQNPELNYVVLMHNGSFNSTRPYQVTLTCSLIILKFPFDTQMCNLSVASFLYPVTDFVMKTRRTPAEIMEDSRSFILTDGEWKFTNLSIVEFTAMMDDKGFSVVTYVISMERRPTLYVLNLILPTCALYLLDMAVLFGPSSLEEKINFQIAIILGSSMLAVILNNSLPTSSNKPPIIVVFFLGTFLLMIMAVLDTFFLLYQQRKSLRLDKVLRSFQQDPQELPKRPMGTLAKGGPQLLPPPKKAQGQGQLTKRLWQLQELDPFLPVLEKVLLFSHLFLSLIFFTVVSIKWSS