Reaction Details Report a problem with these data
Target
D(3) dopamine receptor
Ligand
BDBM82517
Substrate
n/a
Ki
9.3±n/a nM
Comments
PDSP_1289
Citation
Mos, J; Van Hest, A; Van Drimmelen, M; Herremans, AH; Olivier, B The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons. Eur J Pharmacol 325:145-53 (1997) [PubMed] Article
More Info.:
Target
Name:
D(3) dopamine receptor
Synonyms:
DOPAMINE D3 | DRD3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47809.00
Organism:
pigeon
Description:
DOPAMINE D3 DRD3 pigeon::A0A1V4J3K6
Residue:
425
Sequence:
MALFTRSSSHPNTTDPLPCGADNTTESDLPHSHAYYALCYCVLILAIIFGNVLVCLAVLRERTLQTTTNYLVVSLAVADLLVAILVMPWVVYLEVTGGVWTFSRICCDIFVTMDVMMCTASILNLCAISIDRYTAVVKPVQYQYSTGQSSCRRVSLMIVIVWMLAFAVSCPLLFGFNTTGDPSVCSISNPSFVIYSSLVSFYLPFMVTLLLYVRIYLVLRQRQKKRTLTRQGSHSASTKPCYAHKEHMEKKALPNRCQGTSSPCLPLKCSDQETSTKRKLLTVFSLQRYRSFCHEATLTKAPGTAQHSRLEERRKSMKPGLEVRRLSNGRTMSSLKLAHQQPRLIQLRERKATQMLAIVLGAFIVCWLPFFLIHILNTHCPSCHVSPGLYSASTWLGYVNSALNPIIYTTFNTDFRKAFLKILCC