Reaction Details Report a problem with these data
Target
Leukotriene B4 receptor 2
Ligand
BDBM85082
Substrate
n/a
Ki
190±n/a nM
Comments
PDSP_43
Citation
 Yokomizo, T; Izumi, T; Chang, K; Takuwa, Y; Shimizu, T A G-protein-coupled receptor for leukotriene B4 that mediates chemotaxis. Nature 387:620-4 (1997) [PubMed]  Article 
Target
Name:
Leukotriene B4 receptor 2
Synonyms:
BLT2R | BLTR2 | LT4R2_HUMAN | LTB4 receptor JULF2 | LTB4-R 2 | LTB4-R2 | LTB4R2 | LTB4R2 protein | Leukotriene B4 | Leukotriene B4 R2 | Leukotriene B4 receptor | Leukotriene B4 receptor 2 | Leukotriene B4 receptor BLT2 | Leukotriene b1 | Seven transmembrane receptor BLTR2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37964.86
Organism:
Homo sapiens (Human)
Description:
Leukotriene 2 0 HUMAN::Q9NPC1
Residue:
358
Sequence:
MSVCYRPPGNETLLSWKTSRATGTAFLLLAALLGLPGNGFVVWSLAGWRPARGRPLAATLVLHLALADGAVLLLTPLFVAFLTRQAWPLGQAGCKAVYYVCALSMYASVLLTGLLSLQRCLAVTRPFLAPRLRSPALARRLLLAVWLAALLLAVPAAVYRHLWRDRVCQLCHPSPVHAAAHLSLETLTAFVLPFGLMLGCYSVTLARLRGARWGSGRHGARVGRLVSAIVLAFGLLWAPYHAVNLLQAVAALAPPEGALAKLGGAGQAARAGTTALAFFSSSVNPVLYVFTAGDLLPRAGPRFLTRLFEGSGEARGGGRSREGTMELRTTPQLKVVGQGRGNGDPGGGMEKDGPEWDL
  
Inhibitor
Name:
BDBM85082
Synonyms:
20-COOH-LTB4 | CAS_128572 | NSC_128572
Type:
Small organic molecule
Emp. Form.:
C21H32O6
Mol. Mass.:
380.4752
SMILES:
OC(CCCC(O)=O)C=CC=CC=CC(O)CC=CCCCCCC(O)=O |w:18.18,13.13,11.11,9.9|
Structure:
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