Target
Galanin receptor type 2
Ligand
BDBM85163
Substrate
n/a
Ki
840±n/a nM
Comments
PDSP_876
Citation
 Wang, SHashemi, THe, CStrader, CBayne, M Molecular cloning and pharmacological characterization of a new galanin receptor subtype. Mol Pharmacol 52:337-43 (1997) [PubMed]  Article 
Target
Name:
Galanin receptor type 2
Synonyms:
GALR2_RAT | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galnr2 | Galr2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40697.04
Organism:
RAT
Description:
Galanin R2 GALR2 RAT::O08726
Residue:
372
Sequence:
MNGSGSQGAENTSQEGGSGGWQPEAVLVPLFFALIFLVGTVGNALVLAVLLRGGQAVSTTNLFILNLGVADLCFILCCVPFQATIYTLDDWVFGSLLCKAVHFLIFLTMHASSFTLAAVSLDRYLAIRYPLHSRELRTPRNALAAIGLIWGLALLFSGPYLSYYRQSQLANLTVCHPAWSAPRRRAMDLCTFVFSYLLPVLVLSLTYARTLRYLWRTVDPVTAGSGSQRAKRKVTRMIIIVAVLFCLCWMPHHALILCVWFGRFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFRKGFRKICAGLLRPAPRRASGRVSILAPGNHSGSMLEQESTDLTQVSEAAGPLVPPPALPNCTASSRTLDPAC
  
Inhibitor
Name:
BDBM85163
Synonyms:
GMAP (1-41)
Type:
Small organic molecule
Emp. Form.:
C206H327N57O63S
Mol. Mass.:
4642.21
SMILES:
n/a
Structure:
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