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Target
Galanin peptides
Ligand
BDBM85190
Substrate
n/a
Ki
2600±n/a nM
Comments
PDSP_1276
Citation
 Johansson, L; Sohn, D; Thorberg, SO; Jackson, DM; Kelder, D; Larsson, LG; Rényi, L; Ross, SB; Wallsten, C; Eriksson, H; Hu, PS; Jerning, E; Mohell, N; Westlind-Danielsson, A The pharmacological characterization of a novel selective 5-hydroxytryptamine1A receptor antagonist, NAD-299. J Pharmacol Exp Ther 283:216-25 (1997) [PubMed] 
Target
Name:
Galanin peptides
Synonyms:
GALANIN | GALA_RAT | Gal | Galanin peptides | Galn
Type:
Enzyme Catalytic Domain
Mol. Mass.:
13327.23
Organism:
RAT
Description:
GALANIN 0 RAT::P10683
Residue:
124
Sequence:
MARGSVILLAWLLLVATLSATLGLGMPTKEKRGWTLNSAGYLLGPHAIDNHRSFSDKHGLTGKRELPLEVEEGRLGSVAVPLPESNIVRTIMEFLSFLHLKEAGALDSLPGIPLATSSEDLEQS
  
Inhibitor
Name:
BDBM85190
Synonyms:
CAS_3055171 | NAD-299 | NSC_3055171
Type:
Small organic molecule
Emp. Form.:
C18H23FN2O2
Mol. Mass.:
318.3858
SMILES:
NC(=O)c1ccc(F)c2OCC(Cc12)N(C1CCC1)C1CCC1
Structure:
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