Reaction Details Report a problem with these data
Target
Dihydroorotase
Ligand
BDBM85254
Substrate
n/a
Meas. Tech.
Inhibition Assay
pH
7±0
Ki
76000000±0 nM
Citation
Li, Y; Raushel, FM Inhibitors designed for the active site of dihydroorotase. Bioorg Chem 33:470-83 (2005) [PubMed] Article
More Info.:
Target
Name:
Dihydroorotase
Synonyms:
Dihydroorotase (DHO) | PYRC_ECOLI | pyrC
Type:
Enzyme
Mol. Mass.:
38823.92
Organism:
Escherichia coli
Description:
P05020
Residue:
348
Sequence:
MTAPSQVLKIRRPDDWHLHLRDGDMLKTVVPYTSEIYGRAIVMPNLAPPVTTVEAAVAYRQRILDAVPAGHDFTPLMTCYLTDSLDPNELERGFNEGVFTAAKLYPANATTNSSHGVTSIDAIMPVLERMEKIGMPLLVHGEVTHADIDIFDREARFIESVMEPLRQRLTALKVVFEHITTKDAADYVRDGNERLAATITPQHLMFNRNHMLVGGVRPHLYCLPILKRNIHQQALRELVASGFNRVFLGTDSAPHARHRKESSCGCAGCFNAPTALGSYATVFEEMNALQHFEAFCSVNGPQFYGLPVNDTFIELVREEQQVAESIALTDDTLVPFLAGETVRWSVKQ