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Target
Angiotensin-converting enzyme 2
Ligand
BDBM85549
Substrate
n/a
Ki
13.7±n/a nM
Comments
PDSP_1338
Citation
 Handa, RK; Harding, JW; Simasko, SM Characterization and function of the bovine kidney epithelial angiotensin receptor subtype 4 using angiotensin IV and divalinal angiotensin IV as receptor ligands. J Pharmacol Exp Ther 291:1242-9 (1999) [PubMed] 
Target
Name:
Angiotensin-converting enzyme 2
Synonyms:
ACE2 | ACE2_BOVIN | Angiotensin IV
Type:
Enzyme Catalytic Domain
Mol. Mass.:
93046.63
Organism:
BOVINE
Description:
Angiotensin IV 0 BOVINE::Q58DD0
Residue:
804
Sequence:
MTGSFWLLLSLVAVTAAQSTTEEQAKTFLEKFNHEAEDLSYQSSLASWNYNTNITDENVQKMNEARAKWSAFYEEQSRMAKTYSLEEIQNLTLKRQLKALQHSGTSALSAEKSKRLNTILNKMSTIYSTGKVLDPNTQECLALEPGLDDIMENSRDYNRRLWAWEGWRAEVGKQLRPLYEEYVVLENEMARANNYEDYGDYWRGDYEVTGAGDYDYSRDQLMKDVERTFAEIKPLYEQLHAYVRAKLMHTYPSYISPTGCLPAHLLGDMWGRFWTNLYSLTVPFEHKPSIDVTEKMENQSWDAERIFKEAEKFFVSISLPYMTQGFWDNSMLTEPGDGRKVVCHPTAWDLGKGDFRIKMCTKVTMDDFLTAHHEMGHIQYDMAYAAQPYLLRNGANEGFHEAVGEIMSLSAATPHYLKALGLLAPDFHEDNETEINFLLKQALTIVGTLPFTYMLEKWRWMVFKGEIPKQQWMEKWWEMKREIVGVVEPLPHDETYCDPACLFHVAEDYSFIRYYTRTIYQFQFHEALCKTAKHEGALFKCDISNSTEAGQRLLQMLRLGKSEPWTLALENIVGIKTMDVKPLLNYFEPLFTWLKEQNRNSFVGWSTEWTPYSDQSIKVRISLKSALGENAYEWNDNEMYLFQSSVAYAMRKYFSEARNETVLFGEDNVWVSDKKPRISFKFFVTSPNNVSDIIPRTEVENAIRLSRDRINDVFQLDDNSLEFLGIQPTLGPPYEPPVTIWLIIFGVVMGVVVIGIVVLIFTGIRNRRKKNQASSEENPYGSVDLNKGENNSGFQNIDDVQTSL
  
Inhibitor
Name:
BDBM85549
Synonyms:
NleYI-6-hexamide
Type:
Small organic molecule
Emp. Form.:
C21H34N4O3
Mol. Mass.:
390.5197
SMILES:
CCCC[C@H](N)C(=O)N[C@H](Cc1ccccc1)C(=O)NCCCCCC(N)=O |r|
Structure:
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