Reaction Details Report a problem with these data
Target
Hrh3 protein
Ligand
BDBM22542
Substrate
n/a
Ki
1.4±n/a nM
Comments
PDSP_974
Citation
 Lovenberg, TW; Pyati, J; Chang, H; Wilson, SJ; Erlander, MG Cloning of rat histamine H(3) receptor reveals distinct species pharmacological profiles. J Pharmacol Exp Ther 293:771-8 (2000) [PubMed] 
Target
Name:
Hrh3 protein
Synonyms:
HISTAMINE H3 | HRH3 | Hrh3 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37860.96
Organism:
RAT
Description:
Q5PPG3
Residue:
344
Sequence:
MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFVADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCASSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAGPEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDY
  
Inhibitor
Name:
BDBM22542
Synonyms:
4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imidazol-5-ylmethyl)piperidine | Immepip
Type:
Small organic molecule
Emp. Form.:
C9H15N3
Mol. Mass.:
165.2355
SMILES:
C(C1CCNCC1)c1cnc[nH]1
Structure:
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