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Targetadrenergic Alpha2
LigandBDBM81773
Substrate/Competitorn/a
Ki 46±n/a nM
CommentsPDSP_340
Citation Naselsky, DPAshton, DRuffolo, RRHieble, JP Rabbit alpha2-adrenoceptors: both platelets and adipocytes have alpha2A-pharmacology. J Pharmacol Exp Ther298:219-25 (2001) [PubMed]
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adrenergic Alpha2
Name:adrenergic Alpha2
Synonyms:Alpha-2B adrenergic receptor
Type:Enzyme Catalytic Domain
Mol. Mass.:42909.14
Organism:RABBIT
Description:adrenergic Alpha2 0 RABBIT::O77830
Residue:394
Sequence:
AIAAVITFLILFTIFGNALVILAVLTSRSLRAPQNLFLVSLAAADILVATLIIPFSLANE
LLGYWYFRRTWCEVYLALDVLFCTSSIVHLCAISLDRYWAVSRALEYNCKRTPRRIKCII
LTVWLIAAAISLPPLIYKGDQGPQPHGAPQCKLNQEAWYILSSSLGSFFVPCLIMILVYL
RIYLIAKRSHRRGPRAKGGPGEGESRQACPVPGGPSASAKLPTLATPVASASEANGPSKP
AGEKEEGETPEDPGTQALPPGWATLPNSGQGQKEGVSGASLEEEAEEEEEEEEEEDEPQA
VPVSPASVGSPPLQQPQGSRVLATLRGQVLVGRGVGAMSGQWWRRRAQLSREKRFTFVLA
VVIGVFVLCWFPFFFSYSLSAICPQQCRVPHGLF
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  Blast E-value cutoff:
BDBM81773
n/a
NameBDBM81773
Synonyms:BAM 1303 | BAM-1303 | CAS_115219-10-8
TypeSmall organic molecule
Emp. Form.C25H25BrN4
Mol. Mass.461.397
SMILESCN1C[C@H](Cn2ccnc2-c2ccccc2)C[C@H]2[C@H]1Cc1c(Br)[nH]c3cccc2c13 |r|
Structure
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