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Target
Opioid receptor delta 1
Ligand
BDBM86258
Substrate
n/a
Ki
278±n/a nM
Comments
PDSP_1250
Citation
 Gilbert, AK; Hosztafi, S; Mahurter, L; Pasternak, GW Pharmacological characterization of dihydromorphine, 6-acetyldihydromorphine and dihydroheroin analgesia and their differentiation from morphine. Eur J Pharmacol 492:123-30 (2004) [PubMed]  Article 
Target
Name:
Opioid receptor delta 1
Synonyms:
n/a
Type:
PROTEIN
Mol. Mass.:
40708.41
Organism:
Bos taurus
Description:
ChEMBL_863801
Residue:
372
Sequence:
MEPAPSRDPELQPQLLANASEAFPSAFPSAGANASGPPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKVVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPRDGAVVCMLQFPNPSWYWDTVTKICVFLFAFVVPILVITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRMPCGRREPSSFSRAREATARERVTACTPSDGPGGGAAA
  
Inhibitor
Name:
BDBM86258
Synonyms:
CAS_23552-18-3 | Morphine | NSC_5980
Type:
Small organic molecule
Emp. Form.:
C17H19NO3
Mol. Mass.:
285.3377
SMILES:
CN1CCC23C4Oc5c2c(CC1C3C=CC4O)ccc5O |c:16,TLB:13:12:1.2.3:10.9.8|
Structure:
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