Reaction Details Report a problem with these data
Target
GTP-binding nuclear protein GSP2/CNR2
Ligand
BDBM87014
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_8601
Citation
Wang, H; Duffy, RA; Boykow, GC; Chackalamannil, S; Madison, VS Identification of novel cannabinoid CB1 receptor antagonists by using virtual screening with a pharmacophore model. J Med Chem 51:2439-46 (2008) [PubMed] Article
More Info.:
Target
Name:
GTP-binding nuclear protein GSP2/CNR2
Synonyms:
CANNABINOID CB2 | CNR2 | GSP2 | GSP2_YEAST | GTP-binding nuclear protein GSP2/CNR2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
24990.72
Organism:
Saccharomyces cerevisiae
Description:
CANNABINOID CB2 CNR2 0::P32836
Residue:
220
Sequence:
MSAPAQNNAEVPTFKLVLVGDGGTGKTTFVKRHLTGEFEKKYIATIGVEVHPLSFYTNFGEIKFDVWDTAGQEKFGGLRDGYYINAQCAIIMFDVTSRITYKNVPNWHRDLVRVCENIPIVLCGNKVDVKERKVKAKTITFHRKKNLQYYDISAKSNYNFEKPFLWLARKLAGNPQLEFVASPALAPPEVQVDEQLMHQYQQEMDQATALPLPDEDDADL