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Target
Melanocortin receptor 4
Ligand
BDBM88436
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89218±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88436
Synonyms:
MLS000573965 | N-[(6-methyl-2-pyridyl)thiocarbamoyl]-2,2-diphenyl-acetamide | N-[(6-methylpyridin-2-yl)carbamothioyl]-2,2-diphenyl-ethanamide | N-[(6-methylpyridin-2-yl)carbamothioyl]-2,2-diphenylacetamide | N-[[(6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-2,2-diphenylacetamide | N-{[(6-methyl-2-pyridinyl)amino]carbonothioyl}-2,2-diphenylacetamide | SMR000195552 | cid_1224409
Type:
Small organic molecule
Emp. Form.:
C21H19N3OS
Mol. Mass.:
361.46
SMILES:
Cc1cccc(NC(=S)NC(=O)C(c2ccccc2)c2ccccc2)n1
Structure:
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