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Target
Melanocortin receptor 4
Ligand
BDBM88449
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89180±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88449
Synonyms:
4-[9-(4-aminophenyl)-9-fluorenyl]aniline | 4-[9-(4-aminophenyl)-9H-fluoren-9-yl]phenylamine | 4-[9-(4-aminophenyl)fluoren-9-yl]aniline | MLS000584167 | SMR000203330 | [4-[9-(4-aminophenyl)fluoren-9-yl]phenyl]amine | cid_631552
Type:
Small organic molecule
Emp. Form.:
C25H20N2
Mol. Mass.:
348.4397
SMILES:
Nc1ccc(cc1)C1(c2ccccc2-c2ccccc12)c1ccc(N)cc1
Structure:
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