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Target
Melanocortin receptor 4
Ligand
BDBM88498
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89187±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88498
Synonyms:
(4-fluorophenyl)methyl-hexadecyl-dimethyl-azanium;chloride | (4-fluorophenyl)methyl-hexadecyl-dimethylammonium;chloride | (4-fluorophenyl)methyl-hexadecyl-dimethylazanium;chloride | MLS002702413 | SMR001565975 | cetyl-(4-fluorobenzyl)-dimethyl-ammonium;chloride | cid_392616
Type:
Small organic molecule
Emp. Form.:
C25H45FN
Mol. Mass.:
378.6294
SMILES:
CCCCCCCCCCCCCCCC[N+](C)(C)Cc1ccc(F)cc1
Structure:
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