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Target
Melanocortin receptor 4
Ligand
BDBM88608
Substrate
n/a
Meas. Tech.
TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R)
IC50
>64592±n/a nM
Citation
 PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88608
Synonyms:
9,10-diketoanthracene-1-carboxylic acid [2-(2,5-dimethylanilino)-2-keto-ethyl] ester | 9,10-dioxo-1-anthracenecarboxylic acid [2-(2,5-dimethylanilino)-2-oxoethyl] ester | MLS000390666 | SMR000259705 | [2-(2,5-dimethylanilino)-2-oxoethyl] 9,10-dioxoanthracene-1-carboxylate | [2-[(2,5-dimethylphenyl)amino]-2-oxidanylidene-ethyl] 9,10-bis(oxidanylidene)anthracene-1-carboxylate | cid_3503149
Type:
Small organic molecule
Emp. Form.:
C25H19NO5
Mol. Mass.:
413.4221
SMILES:
Cc1ccc(C)c(NC(=O)COC(=O)c2cccc3C(=O)c4ccccc4C(=O)c23)c1
Structure:
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