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Target
Mitochondrial peptide methionine sulfoxide reductase
Ligand
BDBM91490
Substrate
n/a
Meas. Tech.
Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA)
EC50
>103919±n/a nM
Citation
 PubChem, PC Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA) PubChem Bioassay (2012)[AID] 
Target
Name:
Mitochondrial peptide methionine sulfoxide reductase
Synonyms:
MSRA | MSRA protein | MSRA_BOVIN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25822.90
Organism:
Bos taurus
Description:
gi_73586699
Residue:
233
Sequence:
MLSATRRALQLFHSLFPIPRMGDSAAKIVSPQEALPGRKEPLVVAAKHHVNGNRTVEPFPEGTQMAVFGMGCFWGAERKFWTLKGVYSTQVGFAGGYTPNPTYKEVCSGKTGHAEVVRVVFQPEHISFEELLKVFWENHDPTQGMRQGNDHGSQYRSAIYPTSAEHVGAALKSKEDYQKVLSEHGFGLITTDIREGQTFYYAEDYHQQYLSKDPDGYCGLGGTGVSCPLGIKK
  
Inhibitor
Name:
BDBM91490
Synonyms:
1-(8-methyl-1,3,4,5-tetrahydropyrid[4,3-b]indol-2-yl)-2-[4-(2-pyridyl)piperazino]ethanone | 1-(8-methyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)-2-(4-pyridin-2-ylpiperazin-1-yl)ethanone | 1-(8-methyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)-2-[4-(2-pyridinyl)-1-piperazinyl]ethanone | MLS000081152 | SMR000042886 | cid_662231
Type:
Small organic molecule
Emp. Form.:
C23H27N5O
Mol. Mass.:
389.4934
SMILES:
Cc1ccc2[nH]c3CCN(Cc3c2c1)C(=O)CN1CCN(CC1)c1ccccn1
Structure:
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