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TargetKallikrein 14
LigandBDBM113060
Substrate/Competitorn/a
Meas. Tech.KLK14 Assay
pH8±n/a
Temperature310.15±n/a K
Ki 100±n/a nM
Commentsextracted
Citation Wagberg, FLeonardsson, G Benzoxazinone derivatives for treatment of skin diseases US Patent US9695194 Publication Date 7/4/2017
More Info.:Get all data from this article,  Assay Method
 
Kallikrein 14
Name:Kallikrein 14
Synonyms:KLK-L6 | Kallikrein-14 | Kallikrein-like protein 6 | hK14
Type:PROTEIN
Mol. Mass.:29136.99
Organism:Homo sapiens
Description:ChEMBL_1282452
Residue:267
Sequence:
MSLRVLGSGTWPSAPKMFLLLTALQVLAIAMTQSQEDENKIIGGHTCTRSSQPWQAALLA
GPRRRFLCGGALLSGQWVITAAHCGRPILQVALGKHNLRRWEATQQVLRVVRQVTHPNYN
SRTHDNDLMLLQLQQPARIGRAVRPIEVTQACASPGTSCRVSGWGTISSPIARYPASLQC
VNINISPDEVCQKAYPRTITPGMVCAGVPQGGKDSCQGDSGGPLVCRGQLQGLVSWGMER
CALPGYPGVYTNLCKYRSWIEETMRDK
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  Blast E-value cutoff:
BDBM113060
NameBDBM113060
Synonyms:US9695194, 1
TypeSmall organic molecule
Emp. Form.C18H17NO4S
Mol. Mass.343.397
SMILESCCOc1cc2c(cc1OC)nc(oc2=O)-c1ccccc1SC
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
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