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TargetSKiNhead family member (skn-1)
LigandBDBM93847
Substrate/Competitorn/a
IC50 2780±n/a nM
Citation PubChem, PC Dose ResponseConfirmation of SKN-1 Inhibitor hits in a fluorescence ratio assay - Set 2 PubChem Bioassay(2012)[AID]
More Info.:Get all data from this article
 
SKiNhead family member (skn-1)
Name:SKiNhead family member (skn-1)
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:70701.17
Organism:Caenorhabditis elegans
Description:P34707
Residue:623
Sequence:
MGGSSRRQRSTSATRRDDKRRRRQCFSSVADDEEETTSIYGVSSIFIWILATSSLILVIS
SPSSNTSIQSSSYDRITTKHLLDNISPTFKMYTDSNNRNFDEVNHQHQQEQDFNGQSKYD
YPQFNRPMGLRWRDDQRMMEYFMSNGPVETVPVMPILTEHPPASPFGRGPSTERPTTSSR
YEYSSPSLEDIDLIDVLWRSDIAGEKGTRQVAPADQYECDLQTLTEKSTVAPLTAEENAR
YEDLSKGFYNGFFESFNNNQYQQKHQQQQREQIKTPTLEHPTQKAELEDDLFDEDLAQLF
EDVSREEGQLNQLFDNKQQHPVINNVSLSEGIVYNQANLTEMQEMRDSCNQVSISTIPTT
STAQPETLFNVTDSQTVEQWLPTEVVPNDVFPTSNYAYIGMQNDSLQAVVSNGQIDYDHS
YQSTGQTPLSPLIIGSSGRQQQTQTSPGSVTVTATATQSLFDPYHSQRHSFSDCTTDSSS
TCSRLSSESPRYTSESSTGTHESRFYGKLAPSSGSRYQRSSSPRSSQSSIKIARVVPLAS
GQRKRGRQSKDEQLASDNELPVSAFQISEMSLSELQQVLKNESLSEYQRQLIRKIRRRGK
NKVAARTCRQRRTDRHDKMSHYI
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  Blast E-value cutoff:
BDBM93847
NameBDBM93847
Synonyms:MLS001018285 | N-(2-bromanyl-11H-pyrido[1,2-b][2,4]benzodiazepin-6-ylidene)-2,4-dinitro-benzamide | N-(2-bromo-11H-pyrido[1,2-b][2,4]benzodiazepin-6-ylidene)-2,4-dinitro-benzamide | N-(2-bromo-11H-pyrido[1,2-b][2,4]benzodiazepin-6-ylidene)-2,4-dinitrobenzamide | SMR000354560 | cid_2337552
TypeSmall organic molecule
Emp. Form.C20H12BrN5O5
Mol. Mass.482.244
SMILES[O-][N+](=O)c1ccc(C(=O)\N=C2/[N-]c3ccc(Br)c[n+]3Cc3ccccc23)c(c1)[N+]([O-])=O
Structure
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n/a