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Target
Perilipin-1
Ligand
BDBM90719
Substrate
n/a
IC50
1596±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5) PubChem Bioassay (2012)[AID] 
Target
Name:
Perilipin-1
Synonyms:
PERI | PLIN | PLIN1 | PLIN1_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
55988.69
Organism:
Homo sapiens (Human)
Description:
gi_223718203
Residue:
522
Sequence:
MAVNKGLTLLDGDLPEQENVLQRVLQLPVVSGTCECFQKTYTSTKEAHPLVASVCNAYEKGVQSASSLAAWSMEPVVRRLSTQFTAANELACRGLDHLEEKIPALQYPPEKIASELKDTISTRLRSARNSISVPIASTSDKVLGAALAGCELAWGVARDTAEFAANTRAGRLASGGADLALGSIEKVVEYLLPPDKEESAPAPGHQQAQKSPKAKPSLLSRVGALTNTLSRYTVQTMARALEQGHTVAMWIPGVVPLSSLAQWGASVAMQAVSRRRSEVRVPWLHSLAAAQEEDHEDQTDTEGEDTEEEEELETEENKFSEVAALPGPRGLLGGVAHTLQKTLQTTISAVTWAPAAVLGMAGRVLHLTPAPAVSSTKGRAMSLSDALKGVTDNVVDTVVHYVPLPRLSLMEPESEFRDIDNPPAEVERREAERRASGAPSAGPEPAPRLAQPRRSLRSAQSPGAPPGPGLEDEVATPAAPRPGFPAVPREKPKRRVSDSFFRPSVMEPILGRTHYSQLRKKS
  
Inhibitor
Name:
BDBM90719
Synonyms:
4-Bromo-benzoic acid 4-hydroxy-2-(2-oxo-propyl)-naphthalen-1-yl ester | 4-bromobenzoic acid (2-acetonyl-4-hydroxy-1-naphthyl) ester | 4-bromobenzoic acid [4-hydroxy-2-(2-oxopropyl)-1-naphthalenyl] ester | MLS000777412 | SMR000413802 | [4-hydroxy-2-(2-oxopropyl)naphthalen-1-yl] 4-bromobenzoate | [4-oxidanyl-2-(2-oxidanylidenepropyl)naphthalen-1-yl] 4-bromanylbenzoate | cid_2265776
Type:
Small organic molecule
Emp. Form.:
C20H15BrO4
Mol. Mass.:
399.235
SMILES:
CC(=O)Cc1cc(O)c2ccccc2c1OC(=O)c1ccc(Br)cc1
Structure:
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