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Targetnuclear receptor subfamily 5 group A member 2 isoform 2
LigandBDBM54414
Substrate/Competitorn/a
IC50>147.61±n/a nM
Citation PubChem, PC Luminescence-based cell-based high throughput dose response assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) PubChem Bioassay(2013)[AID]
More Info.:Get all data from this article
 
nuclear receptor subfamily 5 group A member 2 isoform 2
Name:Liver Receptor Homolog 1
Synonyms:Alpha-1-fetoprotein transcription factor | B1-binding factor | CYP7A promoter-binding factor | Hepatocytic transcription factor | LRH-1 | Nuclear receptor subfamily 5 group A member 2 | hB1F
Type:Nuclear Hormone Receptor
Mol. Mass.:61341.37
Organism:Homo sapiens (Human)
Description:n/a
Residue:541
Sequence:
MSSNSDTGDLQESLKHGLTPIGAGLPDRHGSPIPARGRLVMLPKVETEALGLARSHGEQG
QMPENMQVSQFKMVNYSYDEDLEELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRY
TCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRALKQ
QKKALIRANGLKLEAMSQVIQAMPSDLTISSAIQNIHSASKGLPLNHAALPPTDYDRSPF
VTSPISMTMPPHGSLQGYQTYGHFPSRAIKSEYPDPYTSSPESIMGYSYMDSYQTSSPAS
IPHLILELLKCEPDEPQVQAKIMAYLQQEQANRSKHEKLSTFGLMCKMADQTLFSIVEWA
RSSIFFRELKVDDQMKLLQNCWSELLILDHIYRQVVHGKEGSIFLVTGQQVDYSIIASQA
GATLNNLMSHAQELVAKLRSLQFDQREFVCLKFLVLFSLDVKNLENFQLVEGVQEQVNAA
LLDYTMCNYPQQTEKFGQLLLRLPEIRAISMQAEEYLYYKHLNGDVPYNNLLIEMLHAKR
A
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BDBM54414
NameBDBM54414
Synonyms:5-Nitro-furan-2-carboxylic acid (4-chloro-benzothiazol-2-yl)-amide | MLS001204059 | N-(4-chloranyl-1,3-benzothiazol-2-yl)-5-nitro-furan-2-carboxamide | N-(4-chloro-1,3-benzothiazol-2-yl)-5-nitro-2-furamide | N-(4-chloro-1,3-benzothiazol-2-yl)-5-nitro-2-furancarboxamide | N-(4-chloro-1,3-benzothiazol-2-yl)-5-nitrofuran-2-carboxamide | SMR000524443 | cid_958637
TypeSmall organic molecule
Emp. Form.C12H6ClN3O4S
Mol. Mass.323.712
SMILES[O-][N+](=O)c1ccc(o1)C(=O)Nc1nc2c(Cl)cccc2s1
Structure
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n/a