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Targetnuclear receptor subfamily 5 group A member 2 isoform 2
LigandBDBM95641
Substrate/Competitorn/a
IC50 4058±n/a nM
Citation PubChem, PC Luminescence-based cell-based high throughput dose response assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) PubChem Bioassay(2013)[AID]
More Info.:Get all data from this article
 
nuclear receptor subfamily 5 group A member 2 isoform 2
Name:Liver Receptor Homolog 1
Synonyms:Alpha-1-fetoprotein transcription factor | B1-binding factor | CYP7A promoter-binding factor | Hepatocytic transcription factor | LRH-1 | Nuclear receptor subfamily 5 group A member 2 | hB1F
Type:Nuclear Hormone Receptor
Mol. Mass.:61341.37
Organism:Homo sapiens (Human)
Description:n/a
Residue:541
Sequence:
MSSNSDTGDLQESLKHGLTPIGAGLPDRHGSPIPARGRLVMLPKVETEALGLARSHGEQG
QMPENMQVSQFKMVNYSYDEDLEELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRY
TCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRALKQ
QKKALIRANGLKLEAMSQVIQAMPSDLTISSAIQNIHSASKGLPLNHAALPPTDYDRSPF
VTSPISMTMPPHGSLQGYQTYGHFPSRAIKSEYPDPYTSSPESIMGYSYMDSYQTSSPAS
IPHLILELLKCEPDEPQVQAKIMAYLQQEQANRSKHEKLSTFGLMCKMADQTLFSIVEWA
RSSIFFRELKVDDQMKLLQNCWSELLILDHIYRQVVHGKEGSIFLVTGQQVDYSIIASQA
GATLNNLMSHAQELVAKLRSLQFDQREFVCLKFLVLFSLDVKNLENFQLVEGVQEQVNAA
LLDYTMCNYPQQTEKFGQLLLRLPEIRAISMQAEEYLYYKHLNGDVPYNNLLIEMLHAKR
A
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BDBM95641
NameBDBM95641
Synonyms:MLS002252657 | N-[2-(1-cyclohexenyl)ethyl]-2-[(2-methyl-8-quinolinyl)oxy]acetamide | N-[2-(cyclohexen-1-yl)ethyl]-2-(2-methylquinolin-8-yl)oxy-ethanamide | N-[2-(cyclohexen-1-yl)ethyl]-2-(2-methylquinolin-8-yl)oxyacetamide | N-[2-(cyclohexen-1-yl)ethyl]-2-[(2-methyl-8-quinolyl)oxy]acetamide | SMR001314994 | cid_2546477
TypeSmall organic molecule
Emp. Form.C20H24N2O2
Mol. Mass.324.4168
SMILESCc1ccc2cccc(OCC(=O)NCCC3=CCCCC3)c2n1 |t:16|
Structure
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n/a