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Target
Trace amine-associated receptor 1
Ligand
BDBM96839
Substrate
n/a
EC50
485.07±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based high throughput dose response assay to identify agonists of the human trace amine associated receptor 1 (TAAR1) PubChem Bioassay (2013)[AID] 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TA1 | TAAR1 | TAAR1_HUMAN | TAR1 | TRAR1 | trace amine-associated receptor 1
Type:
PROTEIN
Mol. Mass.:
39107.47
Organism:
Homo sapiens (Human)
Description:
ChEMBL_792734
Residue:
339
Sequence:
MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNWLIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISIDRYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRGGCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNGISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFNPMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
  
Inhibitor
Name:
BDBM96839
Synonyms:
MLS003270053 | N-[2-(4-hydroxyphenyl)ethyl]-4-phenyl-2-(trifluoromethyl)-1H-imidazole-5-carboxamide | SMR001950448 | cid_51361122
Type:
Small organic molecule
Emp. Form.:
C19H16F3N3O2
Mol. Mass.:
375.3444
SMILES:
Oc1ccc(CCNC(=O)c2[nH]c(nc2-c2ccccc2)C(F)(F)F)cc1
Structure:
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