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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96743
Substrate
n/a
IC50
>29860±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96743
Synonyms:
4-methyl-1,2,3,4-tetrahydro-[1]benzofuro[3,2-c]pyridine;hydrochloride | 4-methyl-1,2,3,4-tetrahydro[1]benzofuro[3,2-c]pyridine | 4-methyl-1,2,3,4-tetrahydrobenzofuro[3,2-c]pyridine;hydrochloride | MLS001180715 | SMR000476894 | cid_12499516
Type:
Small organic molecule
Emp. Form.:
C12H13NO
Mol. Mass.:
187.2377
SMILES:
CC1CNCc2c1oc1ccccc21
Structure:
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