Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM97137
Substrate
n/a
IC50
330.65±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based primary high throughput dose response assay to identify antagonists of the Galanin Receptor 3 (GalR3). PubChem Bioassay (2013)[AID] 
Target
Name:
Galanin receptor type 3
Synonyms:
GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39599.97
Organism:
Homo sapiens (Human)
Description:
Galanin R3 GALR3 HUMAN::O60755
Residue:
368
Sequence:
MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLFILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRARFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHGGEAARGPE
  
Inhibitor
Name:
BDBM97137
Synonyms:
2-Methyl-1-(2-methyl-benzyl)-1H-benzoimidazole | 2-methyl-1-(2-methylbenzyl)benzimidazole | 2-methyl-1-[(2-methylphenyl)methyl]benzimidazole | MLS001211103 | SMR000514923 | cid_2139165
Type:
Small organic molecule
Emp. Form.:
C16H16N2
Mol. Mass.:
236.3116
SMILES:
Cc1nc2ccccc2n1Cc1ccccc1C
Structure:
Search PDB for entries with ligand similarity: