Reaction Details Report a problem with these data
Target
Reverse transcriptase protein
Ligand
BDBM99895
Substrate
n/a
Meas. Tech.
Enzyme Inhibition Assay
IC50
1.128e+4±n/a nM
Citation
Bode, ML; Rousseau, AL; Gravestock, D; Moleele, SS; Van Der Westhuyzen, CW Imidazopyridines and imidazopyrimidines as HIV-1 reverse transcriptase inhibitors US Patent US8501767 Publication Date 8/6/2013
More Info.:
Target
Name:
Reverse transcriptase protein
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
30157.99
Organism:
Human immunodeficiency virus 1
Description:
Q9WJP9
Residue:
259
Sequence:
PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTELEKEGKNSKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNRKTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDKDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLKWGFYTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQK