Reaction Details Report a problem with these data
Target
Gag-Pol polyprotein [484-582,I497V,V499I,E519D,G532V,I538V,R541K,D544E,Q553K,V566A,L573M]
Ligand
BDBM104106
Substrate
n/a
Meas. Tech.
Inhibition Assay
Ki
1.560±0.124 nM
Citation
Shen, Y; Altman, MD; Ali, A; Nalam, MN; Cao, H; Rana, TM; Schiffer, CA; Tidor, B Testing the substrate-envelope hypothesis with designed pairs of compounds. ACS Chem Biol 8:2433-41 (2013) [PubMed] Article
More Info.:
Target
Name:
Gag-Pol polyprotein [484-582,I497V,V499I,E519D,G532V,I538V,R541K,D544E,Q553K,V566A,L573M]
Synonyms:
HIV-1 protease M1 | HIV-1 protease drug-resistant mutant 1 | POL_HV196 | gag-pol
Type:
Protein
Mol. Mass.:
10757.68
Organism:
Human immunodeficiency virus
Description:
Q9QBY3[484-582,I497V,V499I,E519D,G532V,I538V,R541K,D544E,Q553K,V566A,L573M]
Residue:
99
Sequence:
PQITLWQRPIVTVKIGGQLREALLDTGADDTVLEDINLPGKWKPKMIVGIGGFVKVKQYEQVLIEICGKKAIGTVLVGPTPANIIGRNMLTQIGCTLNF