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Target
Adenosine receptor A2
Ligand
BDBM108256
Substrate
n/a
Meas. Tech.
Binding Assay
Ki
951±0.0 nM
Citation
Jagtap, P; Szabo, C; Salzman, AL Purine derivatives as adenosine A1 receptor agonists and methods of use thereof US Patent US8609833 Publication Date 12/17/2013
More Info.:
Target
Name:
Adenosine receptor A2
Synonyms:
ADORA2A | C9JQD8_HUMAN
Type:
Enzyme
Mol. Mass.:
40112.08
Organism:
Homo sapiens (Human)
Description:
C9JQD8
Residue:
365
Sequence:
MPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKNHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMESQPLPGERARSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLRQQEPFKAAGTSARVLAAHGSDGEQVSLRLNGHPPGVWANGSAPHPERRPNGYALGL