Reaction Details Report a problem with these data
Target
Mitogen-activated protein kinase 1
Ligand
BDBM50437407
Substrate
n/a
Meas. Tech.
IMAP-FP Assay
IC50
0.1524±n/a nM
Citation
Lim, J; Kelley, EH; Methot, JL; Zhou, H; Petrocchi, A; Mansoor, UF; Fischer, C; O'Boyle, B; Guerin, DJ; Bienstock, CE; Boyce, CW; Daniels, MH; Falcone, D; Ferguson, RD; Fevrier, S; Huang, X; Lipford, KA; Sloman, DL; Wilson, K; Zhou, W; Witter, D; Maletic, MM; Siliphaivanh, P Compounds that are ERK inhibitors US Patent US9023865 Publication Date 5/5/2015
More Info.:
Target
Name:
Mitogen-activated protein kinase 1
Synonyms:
ERT1 | Erk2 | Extracellular signal-regulated kinase 2 | Extracellular signal-regulated kinase 2 (ERK2) | MAP kinase 1 | MAP kinase 2 | MAP kinase ERK2 | MAPK 1 | MAPK 2 | MK01_MOUSE | Mapk | Mapk1 | Mitogen-activated protein kinase 2 | Prkm1 | p42 | p42-MAPK
Type:
Protein
Mol. Mass.:
41278.65
Organism:
Mus musculus (Mouse)
Description:
P63085
Residue:
358
Sequence:
MAAAAAAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGYRS