Reaction Details Report a problem with these data
Target
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ [1-175]
Ligand
BDBM24777
Substrate
n/a
Meas. Tech.
FabZ Inhibition Assay
pH
7±n/a
Temperature
298.15±n/a K
IC50
5.3e+3± 1.0e+3 nM
Comments
extracted
Citation
McGillick, BE; Kumaran, D; Vieni, C; Swaminathan, S ß-Hydroxyacyl-acyl Carrier Protein Dehydratase (FabZ) from Francisella tularensis and Yersinia pestis: Structure Determination, Enzymatic Characterization, and Cross-Inhibition Studies. Biochemistry 55:1091-9 (2016) [PubMed] Article
More Info.:
Target
Name:
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ [1-175]
Synonyms:
FABZ_YERPY | beta-Hydroxyacyl-acyl carrier protein dehydratase (YpFabZ) | fabZ
Type:
Protein
Mol. Mass.:
19543.64
Organism:
Yersinia pestis
Description:
B1JQH1[1-175]
Residue:
175
Sequence:
MTTDTHTLHIEEILDLLPHRFPFLLVDRVLDFEEGKFLRAVKNVSFNEPFFQGHFPGKPIFPGVLILEAMAQATGILAFKSRGKLEPGELYYFAGIDEARFKRPVVPGDQMIMEVEFVKERRGLTRFTGVAKVDGEIVCTATMMCARSKPAAPAESVVVKPDVVKPDVVNPVVKE