Reaction Details Report a problem with these data
Target
Pantothenate kinase
Ligand
BDBM188489
Substrate
n/a
Meas. Tech.
Biochemical Assay (ATP at Km)
IC50
9e+1±n/a nM
Citation
Björkelid, C; Bergfors, T; Raichurkar, AK; Mukherjee, K; Malolanarasimhan, K; Bandodkar, B; Jones, TA Structural and biochemical characterization of compounds inhibiting Mycobacterium tuberculosis pantothenate kinase. J Biol Chem 288:18260-70 (2013) [PubMed] Article
More Info.:
Target
Name:
Pantothenate kinase
Synonyms:
COAA_MYCTU | Pantothenate kinase (PanK) | coaA
Type:
Protein
Mol. Mass.:
35661.98
Organism:
Mycobacterium tuberculosis ATCC 25618/H37Rv
Description:
n/a
Residue:
312
Sequence:
MSRLSEPSPYVEFDRRQWRALRMSTPLALTEEELVGLRGLGEQIDLLEVEEVYLPLARLIHLQVAARQRLFAATAEFLGEPQQNPDRPVPFIIGVAGSVAVGKSTTARVLQALLARWDHHPRVDLVTTDGFLYPNAELQRRNLMHRKGFPESYNRRALMRFVTSVKSGSDYACAPVYSHLHYDIIPGAEQVVRHPDILILEGLNVLQTGPTLMVSDLFDFSLYVDARIEDIEQWYVSRFLAMRTTAFADPESHFHHYAAFSDSQAVVAAREIWRTINRPNLVENILPTRPRATLVLRKDADHSINRLRLRKL