Reaction Details Report a problem with these data
Target
Lysosomal protective protein [29-480]
Ligand
BDBM193530
Substrate
n/a
Meas. Tech.
Inhibition Assay
pH
5.5±n/a
Temperature
298.15±n/a K
IC50
1390±n/a nM
Comments
extracted
Citation
Ruf, S; Sadowski, T; Wirth, K; Schreuder, H; Buning, C; Kallus, C; Strobel, H; Wehlan, H Biaryl-propionic acid derivatives and their use as pharmaceuticals US Patent US9199947 Publication Date 12/1/2015
More Info.:
Target
Name:
Lysosomal protective protein [29-480]
Synonyms:
CTSA | Cathepsin A | Cathepsin A (CTSA) | PPGB | PPGB_HUMAN
Type:
n/a
Mol. Mass.:
51408.15
Organism:
Homo sapiens (Human)
Description:
P10619[29-480]
Residue:
452
Sequence:
APDQDEIQRLPGLAKQPSFRQYSGYLKGSGSKHLHYWFVESQKDPENSPVVLWLNGGPGCSSLDGLLTEHGPFLVQPDGVTLEYNPYSWNLIANVLYLESPAGVGFSYSDDKFYATNDTEVAQSNFEALQDFFRLFPEYKNNKLFLTGESYAGIYIPTLAVLVMQDPSMNLQGLAVGNGLSSYEQNDNSLVYFAYYHGLLGNRLWSSLQTHCCSQNKCNFYDNKDLECVTNLQEVARIVGNSGLNIYNLYAPCAGGVPSHFRYEKDTVVVQDLGNIFTRLPLKRMWHQALLRSGDKVRMDPPCTNTTAASTYLNNPYVRKALNIPEQLPQWDMCNFLVNLQYRRLYRSMNSQYLKLLSSQKYQILLYNGDVDMACNFMGDEWFVDSLNQKMEVQRRPWLVKYGDSGEQIAGFVKEFSHIAFLTIKGAGHMVPTDKPLAAFTMFSRFLNKQPY