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Target
Bromodomain-containing protein 4 [333-460]
Ligand
BDBM205431
Substrate
n/a
Meas. Tech.
BROMOscan Assay
Kd
0.024±0.0 nM
Citation
Tanaka, M; Roberts, JM; Seo, HS; Souza, A; Paulk, J; Scott, TG; DeAngelo, SL; Dhe-Paganon, S; Bradner, JE Design and characterization of bivalent BET inhibitors. Nat Chem Biol 12:1089-1096 (2016) [PubMed] Article
More Info.:
Target
Name:
Bromodomain-containing protein 4 [333-460]
Synonyms:
BET bromodomain 4(2) (BRD4(2)) | BRD4 | BRD4_HUMAN | Bromodomain-containing protein 4 (BRD4) | HUNK1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
14818.38
Organism:
Homo sapiens (Human)
Description:
aa (333-460)
Residue:
128
Sequence:
KDVPDSQQHPAPEKSSKVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMPDE