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Target
C-terminal-binding protein 1 [A52D]
Ligand
BDBM213227
Substrate
n/a
Meas. Tech.
Equilibrium Dialysis
Kd
5e+2±n/a nM
Citation
Madison, DL; Wirz, JA; Siess, D; Lundblad, JR Nicotinamide adenine dinucleotide-induced multimerization of the co-repressor CtBP1 relies on a switching tryptophan. J Biol Chem 288:27836-48 (2013) [PubMed] Article
More Info.:
Target
Name:
C-terminal-binding protein 1 [A52D]
Synonyms:
C-terminal binding protein (CtBP1 A52D) | CTBP | CTBP1 | CTBP1_HUMAN
Type:
Protein
Mol. Mass.:
47580.80
Organism:
Homo sapiens (Human)
Description:
Human CtBP1 A52D mutant
Residue:
440
Sequence:
MGSSHLLNKGLPLGVRPPIMNGPLHPRPLVALLDGRDCTVEMPILKDVATVDFCDAQSTQEIHEKVLNEAVGALMYHTITLTREDLEKFKALRIIVRIGSGFDNIDIKSAGDLGIAVCNVPAASVEETADSTLCHILNLYRRATWLHQALREGTRVQSVEQIREVASGAARIRGETLGIIGLGRVGQAVALRAKAFGFNVLFYDPYLSDGVERALGLQRVSTLQDLLFHSDCVTLHCGLNEHNHHLINDFTVKQMRQGAFLVNTARGGLVDEKALAQALKEGRIRGAALDVHESEPFSFSQGPLKDAPNLICTPHAAWYSEQASIEMREEAAREIRRAITGRIPDSLKNCVNKDHLTAATHWASMDPAVVHPELNGAAYRYPPGVVGVAPTGIPAAVEGIVPSAMSLSHGLPPVAHPPHAPSPGQTVKPEADRDHASDQL