Reaction Details Report a problem with these data
Target
Orotate phosphoribosyltransferase
Ligand
BDBM214791
Substrate
n/a
Meas. Tech.
Inhibition Assay
pH
8±n/a
Temperature
298.15±n/a K
Ki
220±80 nM
Comments
extracted
Citation
Zhang, Y; Evans, GB; Clinch, K; Crump, DR; Harris, LD; Fröhlich, RF; Tyler, PC; Hazleton, KZ; Cassera, MB; Schramm, VL Transition state analogues of Plasmodium falciparum and human orotate phosphoribosyltransferases. J Biol Chem 288:34746-54 (2013) [PubMed] Article
More Info.:
Target
Name:
Orotate phosphoribosyltransferase
Synonyms:
Orotate phosphoribosyltransferase (PfOPRT)
Type:
Enzyme
Mol. Mass.:
33007.07
Organism:
Plasmodium falciparum
Description:
Q8I3Y0
Residue:
281
Sequence:
MTTIKENEFLCDEEIYKSFVHLKDKICEERKKKELVNNNIDNVNFNDDDDNNYDDDGNSYSSYIKEMKKLLKVVLLKYKALKFGEFILKSKRKSNYFFSSGVLNNIVSSNIICFLLSELILKNKLSFDYLLGASYKGIPMVSLTSHFLFESKKYSNIFYLYDRKEKKEYGDKNVIVGNLDDDDKDILNLKKKTKNNQDEEKKNIIIIDDVFTCGTALTEILAKLKTYEHLKVVAFIVLLNRNEYEINENNQKIYFKDIFEKRVGIPLYSILSYKDDIQSMI