Reaction Details Report a problem with these data
Target
Trans-sialidase [3-643,D247A]
Ligand
BDBM217358
Substrate
n/a
Meas. Tech.
Diffusion Ordered Spectroscopy (DOSY)
Temperature
284.15±n/a K
Kd
1.07e+5± 2e+3 nM
Comments
extracted
Citation
Oliveira, IA; Gonçalves, AS; Neves, JL; von Itzstein, M; Todeschini, AR Evidence of ternary complex formation in Trypanosoma cruzi trans-sialidase catalysis. J Biol Chem 289:423-36 (2014) [PubMed] Article
More Info.:
Target
Name:
Trans-sialidase [3-643,D247A]
Synonyms:
trans-Sialidase (TS D247A)
Type:
Enzyme
Mol. Mass.:
70266.23
Organism:
Trypanosoma cruzi
Description:
T. cruzi TS D247A mutant
Residue:
641
Sequence:
APGSSRVELFKRKNSTVPFEDKAGKVTERVVHSFRLPALVNVDGVMVAIADARYDTSNDNSLIDTVAKYSVDDGETWETQIAIKNSRVSSVSRVVDPTVIVKGNKLYVLVGSYYSSRSYWSSHGDARDWDILLAVGEVTKSIAGGKITASIKWGSPVSLKKFFPAEMEGMHTNQFLGGAGVAIVASNGNLVYPVQVTNKRKQVFSKIFYSEDDGKTWKFGKGRSDFGCSEPVALEWEGKLIINTRVAWKRRLVYESSDMGNTWVEAVGTLSRVWGPSPKSDHPGSQSSFTAVTIEGMRVMLFTHPLNFKGRWLRDRLNLWLTDNQRIYNVGQVSIGDENSAYSSVLYKDDKLYCLHEINTDEVYSLVFARLVGELRIIKSVLRSWKNWDSHLSSICTPADPAASSSESGCGPAVTTVGLVGFLSGNASQNVWEDAYRCVNASTANAERVRNGLKFAGVGGGALWPVSQQGQNQRYRFANHAFTLVASVTIHEAPRAASPLLGASLDSSGGKKLLGLSYDEKHQWQPIYGSTPVTPTGSWETGKRYHVVLTVANKIGSVYIDGELLEGSGQTVVPDGRTPDISHFYVGGYGRSDMPTISHVTVNNVLLYNRQLNTEEIRTLFLSQDLIGTEAHMDSSSDTSA