Reaction Details Report a problem with these data
Target
Ubiquitin carboxyl-terminal hydrolase 2 [258-605]
Ligand
BDBM223976
Substrate
n/a
Meas. Tech.
Di-UB K63-2 Hydrolysis Assay
IC50
3.7e+3± 8e+2 nM
Citation
Magiera, K; Tomala, M; Kubica, K; De Cesare, V; Trost, M; Zieba, BJ; Kachamakova-Trojanowska, N; Les, M; Dubin, G; Holak, TA; Skalniak, L Lithocholic Acid Hydroxyamide Destabilizes Cyclin D1 and Induces G0/G1 Arrest by Inhibiting Deubiquitinase USP2a. Cell Chem Biol 24:458-470 (2017) [PubMed] Article
More Info.:
Target
Name:
Ubiquitin carboxyl-terminal hydrolase 2 [258-605]
Synonyms:
UBP2_HUMAN | UBP41 | USP2 | Ubiquitin-specific peptidase 2a (USP2a)
Type:
Enzyme
Mol. Mass.:
40094.16
Organism:
Homo sapiens (Human)
Description:
Hman USP2a (258-605 aa)
Residue:
348
Sequence:
MNSKSAQGLAGLRNLGNTCFMNSILQCLSNTRELRDYCLQRLYMRDLHHGSNAHTALVEEFAKLIQTIWTSSPNDVVSPSEFKTQIQRYAPRFVGYNQQDAQEFLRFLLDGLHNEVNRVTLRPKSNPENLDHLPDDEKGRQMWRKYLEREDSRIGDLFVGQLKSSLTCTDCGYCSTVFDPFWDLSLPIAKRGYPEVTLMDCMRLFTKEDVLDGDEKPTCCRCRGRKRCIKKFSIQRFPKILVLHLKRFSESRIRTSKLTTFVNFPLRDLDLREFASENTNHAVYNLYAVSNHSGTTMGGHYTAYCRSPGTGEWHTFNDSSVTPMSSSQVRTSDAYLLFYELASPPSRM