Reaction Details Report a problem with these data
Target
Platelet-derived growth factor subunit B
Ligand
BDBM234582
Substrate
n/a
Meas. Tech.
Kinase Assay
pH
7.4±n/a
IC50
16±n/a nM
Comments
extracted
Citation
Boral, S; Malone, TC; Wang, S Indole-1-carboxamides as kinase inhibitors US Patent US9353093 Publication Date 5/31/2016
More Info.:
Target
Name:
Platelet-derived growth factor subunit B
Synonyms:
PDGF | PDGF2 | PDGFB | PDGFB_HUMAN | Platelet-derived growth factor subunit B | Platelet-derived growth factor subunit B (PDGFB) | SIS
Type:
Enzyme
Mol. Mass.:
27298.80
Organism:
Homo sapiens (Human)
Description:
P01127
Residue:
241
Sequence:
MNRCWALFLSLCCYLRLVSAEGDPIPEELYEMLSDHSIRSFDDLQRLLHGDPGEEDGAELDLNMTRSHSGGELESLARGRRSLGSLTIAEPAMIAECKTRTEVFEISRRLIDRTNANFLVWPPCVEVQRCSGCCNNRNVQCRPTQVQLRPVQVRKIEIVRKKPIFKKATVTLEDHLACKCETVAAARPVTRSPGGSQEQRAKTPQTRVTIRTVRVRRPPKGKHRKFKHTHDKTALKETLGA