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TargetFatty acid-binding protein 4 (FABP4)
LigandBDBM234701
Substrate/Competitorn/a
Meas. Tech.Time Resolved-Fluorescence Energy Transfer (TR-FRET) Assay
pH7.5±n/a
IC50 11±n/a nM
Commentsextracted
Citation Buettelmann, BCeccarelli, SMKuehne, HKuhn, BNeidhart, WObst Sander, URichter, H Non-annulated thiophenylamides US Patent US9353102 Publication Date 5/31/2016
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein 4 (FABP4)
Name:Fatty acid-binding protein 4 (FABP4)
Synonyms:A-FABP | AFABP | ALBP | Adipocyte lipid-binding protein | Fatty acid binding protein adipocyte | Fatty acid-binding protein 4
Type:Enzyme
Mol. Mass.:14719.23
Organism:Homo sapiens (Human)
Description:P15090
Residue:132
Sequence:
MCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKN
TEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVM
KGVTSTRVYERA
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  Blast E-value cutoff:
BDBM234701
NameBDBM234701
Synonyms:US9353102, 4.7
TypeSmall organic molecule
Emp. Form.C18H19N3O3S2
Mol. Mass.389.492
SMILESCc1sc(NC(=O)C2=C(CCC2)C(O)=O)c(c1C)-c1nc(ns1)C1CC1 |t:7|
Structure
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