Reaction Details Report a problem with these data
Target
Vascular endothelial growth factor receptor 2 [790-1356]
Ligand
BDBM235397
Substrate
n/a
Meas. Tech.
Inhibition Assay
Temperature
303.15±n/a K
IC50
5.7±n/a nM
Comments
extracted
Citation
More Info.:
Target
Name:
Vascular endothelial growth factor receptor 2 [790-1356]
Synonyms:
FLK1 | KDR | VEGFR2 | VGFR2_HUMAN | Vascular endothelial growth factor receptor 2 (KDR)(790-1356) | Vascular endothelial growth factor receptor 2 (VEGFR2)
Type:
Enzyme
Mol. Mass.:
63329.82
Organism:
Homo sapiens (Human)
Description:
P35968[790-1356]
Residue:
567
Sequence:
KRANGGELKTGYLSIVMDPDELPLDEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKTKGARFRQGKDYVGAIPVDLKRRLDSITSSQSSASSGFVEEKSLSDVEEEEAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDGKDYIVLPISETLSMEEDSGLSLPTSPVSCMEEEEVCDPKFHYDNTAGISQYLQNSKRKSRPVSVKTFEDIPLEEPEVKVIPDDNQTDSGMVLASEELKTLEDRTKLSPSFGGMVPSKSRESVASEGSNQTSGYQSGYHSDDTDTTVYSSEEAELLKLIEIGVQTGSTAQILQPDSGTTLSSPPV