Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM235946
Substrate
n/a
Meas. Tech.
Competition Binding Assay
pH
7.4±n/a
Temperature
303.15±n/a K
Ki
704±n/a nM
Comments
extracted
Citation
 Mechoulam, R; Magid, L; Shohami, E; Bab, I Arylated camphenes, processes for their preparation and uses thereof US Patent  US9365534 Publication Date 6/14/2016 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Homo sapiens (Human)
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM235946
Synonyms:
US9365534, HU-971
Type:
Small Organic Molecule
Emp. Form.:
C24H34O4
Mol. Mass.:
386.5244
SMILES:
CCCCCc1cc(OC)c(C2=C[C@@H]3CC[C@@]2(C(=O)OC)C3(C)C)c(OC)c1 |t:11,THB:10:11:21:14.15|
Structure:
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