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Target
Cannabinoid receptor 1
Ligand
BDBM235937
Substrate
n/a
Meas. Tech.
cAMP Assay
pH
7.5±n/a
Temperature
310.15±n/a K
IC50
3370±n/a nM
Comments
extracted
Citation
 Mechoulam, R; Magid, L; Shohami, E; Bab, I Arylated camphenes, processes for their preparation and uses thereof US Patent  US9365534 Publication Date 6/14/2016 
Target
Name:
Cannabinoid receptor 1
Synonyms:
CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | CNR1_HUMAN | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain)
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
52868.96
Organism:
Homo sapiens (Human)
Description:
P21554
Residue:
472
Sequence:
MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQEKMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIAVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVFHRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLMWTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWKAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLLAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQPLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
  
Inhibitor
Name:
BDBM235937
Synonyms:
US9365534, HU-912
Type:
Small Organic Molecule
Emp. Form.:
C28H42O4
Mol. Mass.:
442.6307
SMILES:
CCCCCCC(C)(C)c1cc(OC)c(C2=C[C@H]3CC[C@]2(C(=O)OC)C3(C)C)c(OC)c1 |t:15,THB:14:15:25:18.19|
Structure:
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