Reaction Details Report a problem with these data
Target
E3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G]
Ligand
BDBM242810
Substrate
n/a
Meas. Tech.
TR-FRET Assay
pH
7.5±n/a
Temperature
310.15±n/a K
IC50
10±n/a nM
Comments
extracted
Citation
Donnell, AF; Kester, R; Lou, Y; Anthony, J; Remiszewski, S 2-oxo-2,3,4,5-tetrahydro-1 H-benzo[B]diazepines and their use in the treatment of cancer US Patent US9422331 Publication Date 8/23/2016
More Info.:
Target
Name:
E3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G]
Synonyms:
API3 | BIRC4 | E3 ubiquitin-protein ligase XIAP (BIR2) | IAP3 | XIAP | XIAP_HUMAN
Type:
Enzyme
Mol. Mass.:
14676.71
Organism:
Artificial Organism
Description:
P98170[124-214,C202A,C213G]
Residue:
125
Sequence:
MRHHHHHHRDHFALDRPSETHADYLLRTGQVVDISDTIYPRNPAMYSEEARLKSFQNWPDYAHLTPRELASAGLYYTGIGDQVQCFACGGKLKNWEPGDFPNCFFVLGRAWSEHRRHRNLNIRSE