Reaction Details Report a problem with these data
Target
Bromodomain-containing protein 4 [352-457]
Ligand
BDBM245909
Substrate
n/a
Meas. Tech.
Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) Assay
pH
6±n/a
Temperature
298.15±n/a K
Ki
17.3±n/a nM
Comments
extracted
Citation
Bogdan, A; Kati, WM; McDaniel, KF; Park, CH; Sheppard, GS; Wang, L Bromodomain inhibitors US Patent US9428514 Publication Date 8/30/2016
More Info.:
Target
Name:
Bromodomain-containing protein 4 [352-457]
Synonyms:
BRD4 | BRD4_HUMAN | Bromodomain-containing protein 4 (BRD4) | Bromodomain-containing protein 4 (BRD4)(aa 352-457) | Bromodomain-containing protein 4 (BRD4-BD2) | HUNK1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12432.37
Organism:
Homo sapiens (Human)
Description:
BDII: amino acid E352-M457
Residue:
106
Sequence:
EQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKM